Copper-catalyzed N-H/S-H functionalization: A strategy for the synthesis of benzothiadiazine derivatives

Dogan S. D.

TETRAHEDRON, cilt.73, ss.2217-2224, 2017 (SCI İndekslerine Giren Dergi) identifier identifier

  • Cilt numarası: 73 Konu: 16
  • Basım Tarihi: 2017
  • Doi Numarası: 10.1016/j.tet.2017.02.063
  • Dergi Adı: TETRAHEDRON
  • Sayfa Sayıları: ss.2217-2224


A copper-mediated N-S bond-forming reaction via N-H/S-H activation is described. This reaction occurs under mild conditions with high efficiency, step economy, and tolerates a wide variety of functional groups, providing an efficient means of accessing biologically important 1,2,4-benzothiadiazin-3(4H)-ones. (C) 2017 Elsevier Ltd. All rights reserved.